| GPCRs
: Receptor binding and reporter based functional
assays
Dopamine D1-4
Histamine H1-3
Muscarinic M1,4,5
Neuropeptide Y1,2
Angiotensin - ATII-2
Cannabinoid-CB1, CB2
Opioid μ,δ,κ
Reporter based transactivation assays
c-JUN
ELK1
CREB
ATF2
c-FOS
CHOP
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Enzymes
BACE1
Cathepsins
Caspase 1, 3 ,9
Protein kinase C
Fatty acid amide hydrolase
MAO-A,B
Signal transduction pathways
cAMP signaling
IP3 signaling
Intracellular calcium signaling
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